CAS RN 432001-19-9
CAS RN 432001-19-9
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Medchem Express C188-9, MedChemExpress
MedChemExpress C188-9 (TTI-101) is a STAT3 inhibitor, with a Kd of 4.7 nM. C188-9 inhibits G-CSF-induced STAT3 activation and STAT3-dependent gene expression. C188-9 induces apoptosis in AML cell lines and primary samples and inhibits colony formation by primary AML blasts.
